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Principles in General Pharmaco...
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Principles in General Pharmacology by Ronald J. Tallarida, Robert B. Raffa, Paul McGonigle.
Saved in:
Bibliographic Details
Main Authors:
Tallarida, Ronald J.
(Author)
,
Raffa, Robert B.
(Author)
,
McGonigle, Paul
(Author)
Corporate Author:
SpringerLink (Online service)
Format:
eBook
Language:
English
Published:
New York, NY :
Springer New York : Imprint: Springer,
1988.
Edition:
1st ed. 1988.
Series:
Springer Series in Pharmacologic Science,
Springer eBook Collection.
Subjects:
Pharmacology.
Pharmacy.
Electronic resources (E-books)
Online Access:
Click to view e-book
Holy Cross Note:
Loaded electronically.
Electronic access restricted to members of the Holy Cross Community.
Holdings
Description
Table of Contents
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Table of Contents:
1 General Principles: History and Overview
Historical Perspective
Principles
Overview of Pharmacologic Principles
References
2 Dose-Effect Relations
Dose-Effect Graphs: Potency and Efficacy
Antagonists
Quantal (All-or-None) Dose-Response Relations
Additivity and Synergism
References
3 Pharmacokinetics
Absorption
Diffusion
Rate Constant for Absorption
Lipid-Water Partition Coefficient
Transport Mechanisms
Electrochemical Potential
The Liver
Drug Elimination
Volume of Distribution
Clearance
Drug-Protein Binding
Protein Binding and Disease
Renal Excretion
Glomerular Filtration
Urine pH and Clearance
Hepatic Clearance
Intravenous Dosing
Repeated Intravenous Injections
Intravenous Infusion
Absorption and Elimination
Extravascular Multiple Dosing
Time Course of Effect and Drug Receptor Concentration
References
4 Drug Metabolism (Biotransformation)
General Principles
Anatomical Sites of Biotransformation
Biotransformation Reactions
Factors Affecting Drug Metabolism
Biotransformations of Selected Common Drugs
References
5 Introduction to Specific Drug Action and Membrane Surface Phenomena
Nonspecific Drug Action
Specific Drug Action: The Development of the Concept of Receptors
Coated Pits and Coated Vesicles
Membrane Capping
Conclusion
References
6 Drugs and Receptors: Chemical Bonding
General Principles
Types of Bonds
Bond Formation in the Drug-Receptor Interaction
References
Appendix A. Physical Constants
Appendix B. Comparison of Atomic, Ionic, and Hydrated Radii of Some Chemical Elements
Appendix C. Structures of Drug Groups
7 The Rate of Drug-Receptor Interactions
Measuring the Rate of Chemical Reactions
Rates of Equilibrium Reactions
Rate of the Drug-Receptor Interaction
Influence of Diffusion on Reaction Rate
Suggested Reading
8 Pharmacodynamics: The Interaction of Drugs with Receptors
Pharmacologic Receptors
Formation of the Drug-Receptor Complex
Classical Theory
Alterations in Classical Drug-Receptor Theory and Alternative Approaches
Dissociation Constants
Drug Combinations: Isoboles
A Changing Receptor Concentration: Modification of Rate Equations
References
9 Radioligand Binding
Direct Binding
Analysis of Receptor Subtypes
Radioligand-Binding Techniques
References
Appendix: Mathematical Tables.
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